Compound Monograph

Vasicine

Vasicine is a pyrroloquinazoline alkaloid from Malabar nut, known for bronchodilator and respiratory effects.

Classification

Vasicine is a pyrroloquinazoline alkaloid, part of the alkaloids class. Nitrogen-containing, often bitter and physiologically potent compounds — the group behind many of the strongest plant medicines and poisons.

Where Does It Come From? (4)

Vasicine is a naturally occurring pyrroloquinazoline alkaloid, found in Malabar nut, Wireweed and 2 other sources. It is flagged as moderately toxic.

Goat's RueMalabar nutSyrian Rue Wireweed Sida acuta

Research & Evidence

Vasicine is a pyrroloquinazoline alkaloid found notably in Malabar nut (Justicia adhatoda), a plant long used in traditional medicine for respiratory complaints. It has documented bronchodilator and respiratory stimulant activity, and it served as a lead structure for the development of the semi-synthetic expectorant bromhexine and its metabolite ambroxol.

Toxicity & Safety

Vasicine has uterotonic (oxytocic) activity and is therefore inappropriate in pregnancy. Its broader safety profile in isolation is only moderately characterised.